3-Bromo-6-iodo-2-methylpyridine

Name: 3-Bromo-6-iodo-2-methylpyridine
Brand: ChemScene
Availability: InStock
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CAS No. 1008361-77-0
Cat. No. CS-0194418
Purity≥96%
MDL No.None

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Type	HazMat Fee
Excepted Quantity	$0.00
FedEx Limited Quantities Ground	$0.00
Hazmat Ground shipping	$50.00+
Inaccessible (Haz class 6.1 or 9), Domestic	$68.00+
Accessible (Haz class 3, 4, 5 or 8), Domestic	$158.00+
Inaccessible (Haz class 6.1 or 9), International	$108.00+
Accessible (Haz class 3, 4, 5 or 8), International	$238.00+

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3-Bromo-6-iodo-2-methylpyridine|CS-0194418

Structure of 1008361-77-0

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General Information

CAS No. 1008361-77-0
Cat. No. CS-0194418
Purity ≥96%
MDL No. None
Storage 4°C, protect from light
Shipping Room temperature in continental US; may vary elsewhere.
Molecular Formula C₆H₅BrIN
Molecular Weight 297.92
Synonym(s) None
SMILES CC1=NC(=CC=C1Br)I

Description

3-Bromo-6-iodo-2-methylpyridine features a sterically accessible pyridine core with complementary halogen handles enabling sequential cross-coupling. The ortho-methyl group enhances regiochemical control, while the bromo and iodo substituents facilitate efficient Pd-catalyzed transformations under standard conditions. This bifunctional scaffold enables rapid access to complex heterocyclic architectures in medicinal chemistry and materials synthesis.

Application

3-Bromo-6-iodo-2-methylpyridine serves as a versatile building block in transition-metal-catalyzed cross-coupling reactions, enabling sequential functionalization of heteroaromatic scaffolds. The ortho-bromo and para-iodo substituents provide complementary reactivity for Pd- or Ni-catalyzed coupling protocols, while the methyl group offers a handle for further derivatization. Its bench-stable nature and high regioselectivity facilitate efficient synthesis of complex pyridine-based architectures relevant to medicinal chemistry and materials science.

Synthesis

Route1
- In-stock
  
  39919-65-8
- ~71%
- In-stock
  
  1008361-77-0
References
- ALMIRALL, S.A.; DRACONIS PHARMA, S.L.; LABORATORIOS DEL DR. ESTEVE, S.A.; AGUILAR, Nuria; FERNANDEZ, Joan, Carles; TERRICABRAS, Emma; CARCELLER GONZALEZ, Elena; GARCIA GARCIA, Francisco, Javier; SALAS SOLANA, Jordi Patent: WO2013/149996 A1, 2013 ; Location in patent: Page/Page column 68 ;

Safety Information

Download SDS

GHS Pictogram :	GHS No : GHS07
Signal Word : Warning	UN#: N/A
Class : N/A	Packing Group : N/A
Hazard Statements : H302-H315-H320-H335
Precautionary Statements : P261-P302+P352

Quality Control

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Computational Chemistry Data

TPSA 12.89
LogP 2.75712
H_Acceptors 1
H_Donors 0
Rotatable_Bonds 0

Other Classifications

Building Blocks Functional Group Bromide

Building Blocks Skeleton Aromatic heterocycle compounds Pyridine compounds

Key Words

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3-Bromo-6-iodo-2-methylpyridine

CAS No. 1008361-77-0

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