4-Bromo-N-methyl-2-pyrimidinamine

Name: 4-Bromo-N-methyl-2-pyrimidinamine
Brand: ChemScene
Availability: InStock
Rating: 5 (1 reviews)

CAS No. 1209458-16-1
Cat. No. CS-W009033
Purity≥98%
MDL No.MFCD13193672

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Type	HazMat Fee
Excepted Quantity	$0.00
FedEx Limited Quantities Ground	$0.00
Hazmat Ground shipping	$50.00+
Inaccessible (Haz class 6.1 or 9), Domestic	$68.00+
Accessible (Haz class 3, 4, 5 or 8), Domestic	$158.00+
Inaccessible (Haz class 6.1 or 9), International	$108.00+
Accessible (Haz class 3, 4, 5 or 8), International	$238.00+

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4-Bromo-N-methyl-2-pyrimidinamine|CS-W009033

Structure of 1209458-16-1

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Description

4-Bromo-N-methyl-2-pyrimidinamine features a bromine substituent at the 4-position and a methylamino group at nitrogen-2, creating a versatile scaffold for medicinal chemistry. The electron-deficient pyrimidine core enables efficient coupling reactions, while the N-methyl group enhances metabolic stability and membrane permeability. This compound serves as a key intermediate in the synthesis of kinase inhibitors and antiviral agents.

Application

4-Bromo-N-methyl-2-pyrimidinamine serves as a versatile building block in medicinal chemistry, enabling palladium-catalyzed cross-coupling reactions due to its reactive bromine and amine functionalities. The N-methyl group enhances metabolic stability while maintaining compatibility with standard coupling protocols. Its pyrimidine core provides a scaffold for constructing bioactive heterocycles, offering bench-stable, easily purified reagents ideal for iterative synthesis workflows in API development.

General Information

CAS No. 1209458-16-1
Cat. No. CS-W009033
Purity ≥98%
MDL No. MFCD13193672
Storage 4°C, protect from light
Shipping Room temperature in continental US; may vary elsewhere.
Molecular Formula C₅H₆BrN₃
Molecular Weight 188.03
Synonym(s) 4-Bromo-N-methylpyrimidin-2-amine
SMILES CNC1=NC=CC(Br)=N1

Computational Chemistry Data

TPSA 37.81
LogP 1.2808
H_Acceptors 3
H_Donors 1
Rotatable_Bonds 1

Safety Information

Download SDS

GHS Pictogram :	GHS No : GHS07
Signal Word : Warning	UN#: N/A
Class : N/A	Packing Group : N/A
Hazard Statements : H302-H315-H319-H335
Precautionary Statements : P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501

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Other Classifications

Building Blocks Functional Group Bromide

Building Blocks Skeleton Aromatic heterocycle compounds Pyrimidine compounds

Key Words

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4-Bromo-N-methyl-2-pyrimidinamine

CAS No. 1209458-16-1

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