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Home   >>   Product   >>  Metabolic Disease
Cat.No. Product Name / Introduction Added
CS-0181 CHIR-99021 August 2016
CHIR-99021 (CT99021) is a GSK-3α/β inhibitor with IC50 of 10 nM/6.
 
CS-0228 GSK1292263 August 2016
GSK1292263 is a novel GPR119 receptor agonist used for the treatment of type 2 diabetes.
 
CS-0277 Odanacatib August 2016
Odanacatib (MK 0822) is a potent, selective, and neutral inhibitor of cathepsin K (human/rabbit) with IC50 of 0.
 
CS-0282 TAK-875 August 2016
TAK-875 is a potent, selective and orally bioavailable GPR40 agonist with EC50 of 0.
 
CS-0289 Taranabant August 2016
Taranabant(MK 0364) is a cannabinoid 1 receptor inverse agonist with IC50 of 0.
 
CS-0300 T863 August 2016
T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA binding site of DGAT1, and inhibits triacylglycerol synthesis in cells.
 
CS-0304 GW_4064 August 2016
GW 4064 is a selective, non-steroidal farnesoid X receptor (FXR) agonist (EC50 = 15 nM).
 
CS-0308 A_922500 August 2016
coe in vivo: Zucker fatty rats and diet-induced dyslipidemic hamsters were dosed orally with A-922500 (0.
 
CS-0316 WAY-362450 August 2016
WAY-362450 (XL335; Turofexorate isopropyl) is a highly potent, selective, and orally active farnesoid X receptor (FXR) agonist with an EC50 of 4 nM.
 
CS-0319 NPS-2143 August 2016
NPS-2143(SB 262470A ) is a selective potent calcium ion-sensing receptor antagonist with IC50 of 43 and 41 nM for cytoplasmic Ca2+ concentrations and parathyroid hormone secretion, respectively.
 
CS-0320 NPS-2143_(hydrochloride) August 2016
NPS-2143(SB 262470A ) is a selective potent calcium ion-sensing receptor antagonist with IC50 of 43 and 41 nM for cytoplasmic Ca2+ concentrations and parathyroid hormone secretion, respectively.
 
CS-0324 MK_0893 August 2016
MK 0893 is a potent, selective glucagon receptor antagonist with IC50 of 6.
 
CS-0325 Etomoxir August 2016
Etomoxir is a cell-permeable, irreversible, and stereospecific inhibitor of carnitine palmitoyltransferase (CPT)-1 and DGAT activity in the mitochondria of rat heart H9c2 myoblastic cells at a concentration of 1-80 μM and 40 μM, respectively.
 
CS-0335 CPA_inhibitor August 2016
CPA inhibitor is a potent inhibitor for carboxypeptidase A (CPA).
 
CS-0365 Fagomine August 2016
D-Fagomine is an iminosugar originally isolated from seeds of buckwheat (Fagopyrum sculentum Moench), present in the human diet and now available as a pure crystalline product.
 
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CS-0645 Rimonabant
Rimonabant(SR141716) is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.
CS-2222 Meprednisone
Meprednisone is a glucocorticoid and a methylated derivative of prednisone.
CS-0264 DAPT
DAPT(GSI-IX) is an inhibitor of γ-secretase; DAPT causes a reduction in Aβ40 and Aβ42 levels in human primary neuronal cultures (IC50 values are 115 and 200 nM for total Aβ and Aβ42 respectively) and in brain extract, cerebrospinal fluid and plasma in vivo.
CS-0613 Tideglusib
Tideglusib(NP-031112) is an irreversible, non ATP-competitive GSK-3β inhibitor with IC50 of 60 nM.
CS-0757 SB-705498
SB-705498 is a potent, selective and orally bioavailable transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with a pIC50 of 7.
CS-0766 Aripiprazole
Aripiprazole(Abilify) is a human 5-HT1A receptor partial agonist with a Ki of 4.
CS-1971 Haloperidol
Haloperidol blocks dopamine receptors in in the treatment of schizophrenia, acute psychosis, and delirium.
CS-0609 SCH 527123
SCH-527123 is a potent antagonist of both CXCR1 and CXCR2 with IC50 of 42 nM and 3 nM, respectively.
CS-0361 Boceprevir
Boceprevir(EBP-520, SCH503034) is an HCV protease inhibitor (Ki=14 nM) for the treatment of hepatitis C virus infection.
CS-0625 Avosentan
Avosentan(Ro 67-0565; SPP-301) is a potent, selective endothelin receptor(ETA receptor) antagonist.
CS-0494 XAV-939
XAV939 is a small molecule and selective Wnt pathway β-catenin-mediated transcription inhibitor and axin stabilizing agent with IC50 of 11 and 4 nM for the inhibition of TNKS1 and TNKS2, respectively.
CS-0592 YM-201636
YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p110α.
CS-0608 BMS-754807
BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.
CS-0627 MEK162
MEK162(ARRY-438162; ARRY-162) is a potent inhibitor of MEK1/2 with IC50 of 12 nM.
CS-0765 CYT387 (sulfate salt)
CYT387 sulfate(momelotinib) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3.
CS-1955 CC-401
CC-401 is a second generation ATP-competitive anthrapyrazolone c-Jun N terminal kinase (JNK) inhibitor with potential antineoplastic activity.
CS-1956 XL413
XL413 is a potent and selective Cdc7 inhibitor with an IC50 of 3.
CS-B0575 1H-Pyrrolo[2,3-b]pyridin-4-amine, 1-methyl-
CS-B0576 1H-Pyrrolo[2,3-b]pyridine-1-carboxylic acid, 4-amino-, 1,1-dimethylethyl ester
CS-B0577 1H-Pyrrolo[2,3-b]pyridin-4-amine, 1-(phenylmethyl)-

 
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